Substance (mean ± SD) | Cmax (ng/ml) | Tmax (hr) | AUC (0-t) (ng*h/ml) | λz (1/hr) | (t1/2)z (hr) | AUC (0-∞) (ng*h/ml) | AUCext (%) | CL (ml/min/kg) | Vz (l/kg) |
---|---|---|---|---|---|---|---|---|---|
Cocaine Pre Selegiline (session 1) | 721 ± 773 | 2.66 ± 1.74 | 2640 ± 55.6 | 0.453 ± 27.9 | 1.71 ± 0.81 | 2680 ± 1470 | 1.40 ± 1.03 | 18.3 ± 6.17 | 2.49 ± 0.88 |
Cocaine With Selegiline (session 2) | 640 ± 332 | 2.27 ± 2.04 | 2360 ± 499 | 0.456 ± 0.09 | 1.57 ± 0.30 | 2400 ± 487 | 1.78 ± 1.87 | 18.0 ± 3.34 | 2.44 ± 0.64 |
Benzoyl-ecgonine Pre Selegiline (session 1) | 1045 ± 180 | 4.79 ± 0.50 | 13000 ± 3030 | 0.0928 ± 0.023 | 8.63 ± 5.36 | 13600 ± 3820 | 3.45 ± 6.45 |  |  |
Benzoyl-ecgonine With Selegiline (session 2) | 957 ± 184 | 5.04 ± 0.65 | 12900 ± 3760 | 0.0971 ± 0.024 | 7.52 ± 1.82 | 13200 ± 4180 | 2.21 ± 2.24 |  |  |